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GW806742X hydrochloride

Glpbio
Catalog No:GC61454-10mM (in 1mL DMSO) CAS No.: MDLNo:C25H23ClF3N7O4S Brand:Glpbio purity: 特性: Purpose:GW806742Xhydrochloride是一种ATP模拟物,是一种有效的MLKL抑制剂,结合MLKL假激酶结构域,Kd值为9.3μM。GW806742Xhydrochloride具有抗VEGFR2的活性(IC50=2nM)。GW806742Xhydrochloride延缓MLKL膜移位并抑制坏死。DMSO: 100 mg/mL (163.93 mM; Need ultrasonic); H2O: < 0.1 mg/mL (ultrasonic) (insoluble)
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